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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7157 | XY1 | Histone Methyltransferase | |
XY1 is a very close analogue of SGC707 (a potent, selective, and non-competitive inhibitor of PRMT3 with IC50 of 31 nM), It is intended to be used as a negative control for SGC707 in studies involving PRMT3 action. | |||
T60612 | Neboglamine hydrochloride | ||
Neboglamine (CR-2249, XY-2401) hydrochloride is a positive modulator of NMDA receptor glycine site with orally active that can be used in the research of schizophrenia [1]. | |||
T74380 | XY-06-007 | ||
XY-06-007, a potent and selective bump-and-hole (B&H) PROTAC BRD4 BD1 L94V degrader, exhibits a DC50, 6 h of 10 nM specifically against BRD4 BD1 L94V without degrading off-targets. It also demonstrates favorable pharmaco... | |||
T83882 | XY-4 | ||
XY-4, a derivative of 1-palmitoyl lysophosphatidic acid (1-palmitoyl LPA094) and an agonist of peroxisome proliferator-activated receptor γ (PPARγ), effectively induces reporter gene expression in RAW 264.7 macrophages h... | |||
T80759 | XY-52 | ||
XY-52 (Compound 32), an ST2 (Stimulation-2) inhibitor, exhibits IC50 values of 5.68 μM and 4.59 μM in the AlphaLISA and HEK-Blue assays, respectively. It promotes proinflammatory T-cell proliferation and diminishes plasm... |